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申 请 号:CN201811027675
专利名称:含有A.terreus次级代谢产物的抗肿瘤制剂及其制备方法
专利权人:浙江海洋大学
交易方式:协议
参考价格: 面议
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名称: | 含有A.terreus次级代谢产物的抗肿瘤制剂及其制备方法 |
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申请号: | CN201811027675 |
申请日期: | 2018-09-04 |
申请人: | 浙江海洋大学 |
发明人: | 黄芳芳; 孙坤来; 张译文; 王斌; 初学梅; 陈荫; 赵玉勤 |
地址: | 316000 浙江省舟山市定海区临城街道海大南路1号 |
主分类号: | A61K31/353 |
分类号: | A61K31/353; A61P35/00; A61P35/02; C12P17/06; C07D311/04; C12R1/66 |
主权项: | |
摘要: | 本发明公开了一种含有Aterreus次级代谢产物的抗肿瘤制剂及其制备方法,抗肿瘤制剂的有效成分为A.terreus次级代谢产物,其制备方法为:向真菌培养基中添加表观遗传修饰调控剂TSA、烟酰胺、二胜肽,发酵培养,分别萃取发酵液、菌丝体,发酵浓缩物经柱色谱、高效液相色谱分离纯化,得Aterreus次级代谢产物。有益效果为:本发明在培养基中添加烟酰胺、二胜肽,与表观遗传修饰调控剂TSA产生协同增益作用,对Aterreus进行表观遗传修饰,并分离得到目标次级代谢产物;本发明制得的含有Aterreus次级代谢产物的抗肿瘤制剂可用于治疗肺癌、乳腺癌、白血病等癌症,具有较好的抗肿瘤效果。 |
start date | end date | title | description | icon | date limit | importance | link | modal |
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2018-11-13 | 公开 | js/timeglider/js/timeglider/icons/verticalLineGray.png | 50 | |||||
2018-12-07 | 实质审查的生效 | js/timeglider/js/timeglider/icons/verticalLineGray.png | 50 |
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#1 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/Application/Home/Controller/PraiseController.class.php(56): Yar_Client->theme_bar('get_bar_id', Array)
#2 [internal function]: Home\Controller\PraiseController->get_bar_id_by_from_id()
#3 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/ThinkPHP/Library/Think/App.class.php(173): ReflectionMethod->invoke(Object(Home\Controller\PraiseController))
#4 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/ThinkPHP/Library/Think/App.class.php(110): Think\App::invokeAction(Object(Home\Controller\PraiseController), 'get_bar_id_by_f...')
#5 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/ThinkPHP/Library/Think/App.class.php(204): Think\App::exec()
#6 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/ThinkPHP/Library/Think/Think.class.php(120): Think\App::run()
#7 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/ThinkPHP/ThinkPHP.php(97): Think\Think::start()
#8 /home/ftp/1520/ipa361_com-20150420-MrH/ipa361.com/mapi/index.php(27): require('/home/ftp/1520/...')
#9 {main}